BDBM50002338 (Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine::10-(2-(1-methylpiperidin-2-yl)ethyl)-2-(methylthio)-10H-phenothiazine::10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine::10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine (thioridazine)::CHEMBL479::MELLARIL::MELLARIL-S::THIORIDAZINE::TP-21::US9504692, Thioridazine
SMILES CSc1ccc2Sc3ccccc3N(CCC3CCCCN3C)c2c1
InChI Key InChIKey=KLBQZWRITKRQQV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 40 hits for monomerid = 50002338
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-Raclopride from human D2 receptor (unknown origin) expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-haloperidol from Dopamine receptor D2 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Compound was tested in vitro for its affinity towards rat striatal Dopamine receptor D2 labeled with [3H]- spiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory against radioligand [3H]spiperone binding to rat striatal Dopamine receptor D2More data for this Ligand-Target Pair